N-stearyl-[Nle17]VIP [Ligand Id: 2271] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| VPAC1 receptor in Human [GtoPdb: 371] [UniProtKB: P32241] | ||||||||
| GtoPdb | inhibition of [125I]-VIP binding to membranes from CHO cells stably expressing the recombinant receptor | - | 8.3 | pIC50 | 5 | nM | IC50 | Eur J Pharmacol (1998) 354: 105-11 [PMID:9726637] |
| VPAC1 receptor in Rat [GtoPdb: 371] [UniProtKB: P30083] | ||||||||
| GtoPdb | inhibition of [125I]-VIP binding to membranes from CHO cells stably expressing the recombinant receptor | - | 8.7 | pIC50 | 2 | nM | IC50 | Eur J Pharmacol (1998) 354: 105-11 [PMID:9726637] |
| VPAC2 receptor in Human [GtoPdb: 372] [UniProtKB: P41587] | ||||||||
| GtoPdb | inhibition of [125I]Ro25 1553 binding to membranes from CHO cells stably expressing the recombinant receptor | - | 9 | pIC50 | 1 | nM | IC50 | Eur J Pharmacol (1998) 354: 105-11 [PMID:9726637] |
| VPAC2 receptor in Rat [GtoPdb: 372] [UniProtKB: P35000] | ||||||||
| GtoPdb | inhibition of [125I]Ro25 1553 binding to membranes from CHO cells stably expressing the recombinant receptor | - | 8.5 | pIC50 | 3 | nM | IC50 | Eur J Pharmacol (1998) 354: 105-11 [PMID:9726637] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
