N-stearyl-[Nle17] neurotensin-(6-11)/VIP-(7-28) [Ligand Id: 2266] activity data from GtoPdb

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  • PAC1 receptor in Human [GtoPdb: 370] [UniProtKB: P41586]
  • This target only has 0 pki data point
  • 0
1 _lig_chart_1 PAC1 receptor Human
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  • VPAC1 receptor in Human [GtoPdb: 371] [UniProtKB: P32241]
  • This target only has 0 pki data point
  • 0
2 _lig_chart_2 VPAC1 receptor Human
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  • VPAC2 receptor in Human [GtoPdb: 372] [UniProtKB: P41587]
  • This target only has 0 pki data point
  • 0
3 _lig_chart_3 VPAC2 receptor Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
PAC1 receptor in Human [GtoPdb: 370] [UniProtKB: P41586]
GtoPdb inhibition of [125I]-PACAP-27 binding to membranes from NIH/3T3 cells stably expressing the recombinant receptor - 7.2 pIC50 65 nM IC50 J Mol Neurosci (2002) 18: 29-35 [PMID:11931347]
VPAC1 receptor in Human [GtoPdb: 371] [UniProtKB: P32241]
GtoPdb inhibition of [125I]-VIP binding to membranes from CHO cells stably expressing the recombinant receptor - 7.5 pIC50 30 nM IC50 J Mol Neurosci (2002) 18: 29-35 [PMID:11931347]
VPAC2 receptor in Human [GtoPdb: 372] [UniProtKB: P41587]
GtoPdb inhibition of [125I]-VIP binding to membranes from CHO cells stably expressing the recombinant receptor - 7.3 pIC50 50 nM IC50 J Mol Neurosci (2002) 18: 29-35 [PMID:11931347]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.