maxadilan [Ligand Id: 2264] activity data from GtoPdb

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  • PAC1 receptor in Human [GtoPdb: 370] [UniProtKB: P41586]
Created with Highcharts 10.3.3ValuesChart context menuPAC1 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human024681012Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
PAC1 receptor in Human [GtoPdb: 370] [UniProtKB: P41586]
GtoPdb calcium influx in CHO cells stably expressing recombinant receptor - 6.2 pEC50 568 nM EC50 Neuropharmacology (2006) 51: 1086-98 [PMID:16930633]
GtoPdb cyclic AMP formation in CHO cells stably expressing recombinant receptor - 10.3 pEC50 0.05 nM EC50 Neuropharmacology (2006) 51: 1086-98 [PMID:16930633]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.