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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| 5-HT2B receptor in Human [GtoPdb: 7] [UniProtKB: P41595] | ||||||||
| GtoPdb | - | - | 8.4 | pKd | - | - | - | Naunyn Schmiedebergs Arch Pharmacol (1998) 357: 17-24 [PMID:9459568] |
| α2A-adrenoceptor in Human [GtoPdb: 25] [UniProtKB: P08913] | ||||||||
| GtoPdb | - | - | 9.5 | pKd | - | - | - |
J Pharmacol Exp Ther (1996) 278: 1215-27 [PMID:8819505]; Mol Pharmacol (1992) 42: 1-5 [PMID:1353247]; Pharmacol Res Perspect (2022) 10: e00936 [PMID:35224877] |
| α2B-adrenoceptor in Human [GtoPdb: 26] [UniProtKB: P18089] | ||||||||
| GtoPdb | - | - | 9.2 | pKd | - | - | - |
J Pharmacol Exp Ther (1996) 278: 1215-27 [PMID:8819505]; Mol Pharmacol (1992) 42: 1-5 [PMID:1353247]; Pharmacol Res Perspect (2022) 10: e00936 [PMID:35224877] |
| α2C-adrenoceptor in Human [GtoPdb: 27] [UniProtKB: P18825] | ||||||||
| GtoPdb | - | - | 9.9 | pKd | - | - | - |
J Pharmacol Exp Ther (1996) 278: 1215-27 [PMID:8819505]; Mol Pharmacol (1992) 42: 1-5 [PMID:1353247]; Pharmacol Res Perspect (2022) 10: e00936 [PMID:35224877] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.