cenacitinib [Ligand Id: 13487] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| tyrosine kinase 2 in Human [GtoPdb: 2269] [UniProtKB: P29597] | ||||||||
| GtoPdb | Binned value determined as inhibition in aJAK1 /TYK2 stimulated STAT1 phosphorylation assay | - | 6 | pIC50 | <1000 | nM | IC50 | US20210139486A1. Tyk2 pseudokinase ligands (2021) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
