BIIB068 [Ligand Id: 11178] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Bruton tyrosine kinase in Human [GtoPdb: 1948] [UniProtKB: Q06187] | ||||||||
| GtoPdb | - | - | 9.52 | pKd | 0.3 | nM | Kd | J Med Chem (2020) 63: 12526-12541 [PMID:32696648] |
| GtoPdb | Biochemical assay measuring enzyme activity inhibition. | - | 9 | pIC50 | 1 | nM | IC50 | J Med Chem (2020) 63: 12526-12541 [PMID:32696648] |
| Janus kinase 2 in Human [GtoPdb: 2048] [UniProtKB: O60674] | ||||||||
| GtoPdb | - | - | 6.34 | pKd | 460 | nM | Kd | J Med Chem (2020) 63: 12526-12541 [PMID:32696648] |
| mitogen-activated protein kinase kinase kinase 19 in Human [GtoPdb: 2076] [UniProtKB: Q56UN5] | ||||||||
| GtoPdb | - | - | 6.89 | pKd | 130 | nM | Kd | J Med Chem (2020) 63: 12526-12541 [PMID:32696648] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
