WM382 [Ligand Id: 11162] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • Plasmodium falciparum plasmepsin X in Plasmodium falciparum [GtoPdb: 3071]
  • Plasmodium falciparum plasmepsin X in Plasmodium falciparum K1 [GtoPdb: 3071]
  • Plasmodium falciparum plasmepsin X in Plasmodium knowlesi [GtoPdb: 3071]
  • Plasmodium falciparum plasmepsin X in Plasmodium falciparum 3D7 [GtoPdb: 3071] [UniProtKB: Q8IAS0]
  • Plasmodium falciparum plasmepsin X in Plasmodium falciparum Dd2 [GtoPdb: 3071]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Plasmodium falciparum plasmepsin X in Plasmodium falciparum [GtoPdb: 3071]
GtoPdb Peptide cleavage assay using recombinant PMX - 10.46 pKi 0.04 nM Ki Cell Host Microbe (2020) 27: 642-658.e12 [PMID:32109369]
Plasmodium falciparum plasmepsin X in Plasmodium falciparum K1 [GtoPdb: 3071]
GtoPdb Parasite growth inhibition assay - 9.19 pEC50 0.65 nM EC50 Cell Host Microbe (2020) 27: 642-658.e12 [PMID:32109369]
Plasmodium falciparum plasmepsin X in Plasmodium knowlesi [GtoPdb: 3071]
GtoPdb Parasite growth inhibition assay - 9.74 pEC50 0.18 nM EC50 Cell Host Microbe (2020) 27: 642-658.e12 [PMID:32109369]
Plasmodium falciparum plasmepsin X in Plasmodium falciparum 3D7 [GtoPdb: 3071] [UniProtKB: Q8IAS0]
GtoPdb Parasite growth inhibition assay - 9.22 pEC50 0.6 nM EC50 Cell Host Microbe (2020) 27: 642-658.e12 [PMID:32109369]
Plasmodium falciparum plasmepsin X in Plasmodium falciparum Dd2 [GtoPdb: 3071]
GtoPdb Parasite growth inhibition assay - 9.59 pEC50 0.26 nM EC50 Cell Host Microbe (2020) 27: 642-658.e12 [PMID:32109369]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.