WEHI-842 [Ligand Id: 10616] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL3782104
  • Plasmodium falciparum plasmepsin V in Plasmodium falciparum NF54 [GtoPdb: 3106]
  • Plasmodium falciparum plasmepsin V in Plasmodium falciparum 3D7 [GtoPdb: 3106] [UniProtKB: Q8I6Z5]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Plasmodium falciparum plasmepsin V in Plasmodium falciparum NF54 [GtoPdb: 3106]
GtoPdb Parasite gametocyte assay - 7.4 pEC50 40 nM EC50 Cell Rep (2019) 29: 3796-3806.e4 [PMID:31851913]
Plasmodium falciparum plasmepsin V in Plasmodium falciparum 3D7 [GtoPdb: 3106] [UniProtKB: Q8I6Z5]
GtoPdb - - 6.4 pEC50 400 nM EC50 Nat. Struct. Mol. Biol. (2015) 22: 590-6 [PMID:26214367]

ChEMBL data shown on this page come from version 26:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]