MS432 [Ligand Id: 10563] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| mitogen-activated protein kinase kinase 1 in Human [GtoPdb: 2062] [UniProtKB: Q02750] | ||||||||
| GtoPdb | Determined in an in vitro biochemical assay, using a kinase-dead ERK mutant as the substrate for hMEK1. | - | 5.82 | pIC50 | 1500 | nM | IC50 | J Med Chem (2019) 62: 10897-10911 [PMID:31730343] |
| mitogen-activated protein kinase kinase 2 in Human [GtoPdb: 2063] [UniProtKB: P36507] | ||||||||
| GtoPdb | Determined in an in vitro biochemical assay, using a kinase-dead ERK mutant as the substrate for hMEK2. | - | 6.23 | pIC50 | 590 | nM | IC50 | J Med Chem (2019) 62: 10897-10911 [PMID:31730343] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
