elexacaftor [Ligand Id: 10552] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| CFTR in Human [GtoPdb: 707] [UniProtKB: P13569] | ||||||||
| GtoPdb | - | - | 7.15 | pEC50 | 70 | nM | EC50 |
N Engl J Med (2018) 379: 1612-1620 [PMID:30334692]; WO2018107100A1. Modulator of cystic fibrosis transmembrane conductance regulator, pharmaceutical compositions, methods of treatment, and process for making the modulator (2018) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
