THAL-SNS-032 [Ligand Id: 10547] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| cyclin dependent kinase 1 in Human [GtoPdb: 1961] [UniProtKB: P06493] | ||||||||
| GtoPdb | Biochemical inhibition of CDK1/CycB. | - | 6.77 | pIC50 | 171 | nM | IC50 | Nat Chem Biol (2018) 14: 163-170 [PMID:29251720] |
| cyclin dependent kinase 2 in Human [GtoPdb: 1973] [UniProtKB: P24941] | ||||||||
| GtoPdb | Biochemical inhibition of CDK2/cyclin A | - | 7.21 | pIC50 | 62 | nM | IC50 | Nat Chem Biol (2018) 14: 163-170 [PMID:29251720] |
| cyclin dependent kinase 7 in Human [GtoPdb: 1979] [UniProtKB: P50613] | ||||||||
| GtoPdb | Inhibition of CDK7/CycH/MNAT1. | - | 6.4 | pIC50 | 398 | nM | IC50 | Nat Chem Biol (2018) 14: 163-170 [PMID:29251720] |
| cyclin dependent kinase 9 in Human [GtoPdb: 1981] [UniProtKB: P50750] | ||||||||
| GtoPdb | Biochemical inhibition of CDK9/CycT1. | - | 8.4 | pIC50 | 4 | nM | IC50 | Nat Chem Biol (2018) 14: 163-170 [PMID:29251720] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
