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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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MET proto-oncogene, receptor tyrosine kinase in Human [GtoPdb: 1815] [UniProtKB: P08581] | ||||||||
GtoPdb | Inhibition of HGF stimulated c-Met phosphorylation in a cell-based assay. | - | 7.92 | pIC50 | 12 | nM | IC50 | WO2007075567A1. Triazolopyridazines as tyrosine kinase modulators (2007) |
GtoPdb | Inhibition of c-Met autophosphorylation measured in a time resolved fluorescence assay (DELFIA). | - | 9 | pIC50 | 1 | nM | IC50 | WO2007075567A1. Triazolopyridazines as tyrosine kinase modulators (2007) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.