PA21A092 [Ligand Id: 10415] activity data from GtoPdb

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  • Plasmodium falciparum non-SERCA-type Ca2+ -transporting P-ATPase in Plasmodium falciparum TM90C2B [GtoPdb: 2971]
  • Plasmodium falciparum non-SERCA-type Ca2+ -transporting P-ATPase in Plasmodium falciparum FCR3 [GtoPdb: 2971]
  • Plasmodium falciparum non-SERCA-type Ca2+ -transporting P-ATPase in Plasmodium falciparum NF54 [GtoPdb: 2971]
  • Plasmodium falciparum non-SERCA-type Ca2+ -transporting P-ATPase in Plasmodium falciparum 3D7 [GtoPdb: 2971] [UniProtKB: A0A143ZZK9]
  • Plasmodium falciparum non-SERCA-type Ca2+ -transporting P-ATPase in Plasmodium falciparum Dd2 [GtoPdb: 2971]
  • Plasmodium falciparum non-SERCA-type Ca2+ -transporting P-ATPase in Plasmodium falciparum HB3 [GtoPdb: 2971]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Plasmodium falciparum non-SERCA-type Ca2+ -transporting P-ATPase in Plasmodium falciparum TM90C2B [GtoPdb: 2971]
GtoPdb Parasite growth inhibition assay - 7.89 pEC50 13 nM EC50 Nat Commun (2014) 5: 5521 [PMID:25422853]
Plasmodium falciparum non-SERCA-type Ca2+ -transporting P-ATPase in Plasmodium falciparum FCR3 [GtoPdb: 2971]
GtoPdb Parasite growth inhibition assay - 7.72 pEC50 19 nM EC50 Nat Commun (2014) 5: 5521 [PMID:25422853]
Plasmodium falciparum non-SERCA-type Ca2+ -transporting P-ATPase in Plasmodium falciparum NF54 [GtoPdb: 2971]
GtoPdb Parasite dual gamete formation assay (DGFA) - 7.13 pEC50 74 nM EC50 Nat Commun (2014) 5: 5521 [PMID:25422853]
GtoPdb Parasite dual gamete formation assay (DGFA) - 7.41 pEC50 39 nM EC50 Nat Commun (2014) 5: 5521 [PMID:25422853]
Plasmodium falciparum non-SERCA-type Ca2+ -transporting P-ATPase in Plasmodium falciparum 3D7 [GtoPdb: 2971] [UniProtKB: A0A143ZZK9]
GtoPdb Parasite growth inhibition assay - 7.74 pEC50 18 nM EC50 Nat Commun (2014) 5: 5521 [PMID:25422853]
Plasmodium falciparum non-SERCA-type Ca2+ -transporting P-ATPase in Plasmodium falciparum Dd2 [GtoPdb: 2971]
GtoPdb Parasite growth inhibition assay - 7.66 pEC50 22 nM EC50 Nat Commun (2014) 5: 5521 [PMID:25422853]
Plasmodium falciparum non-SERCA-type Ca2+ -transporting P-ATPase in Plasmodium falciparum HB3 [GtoPdb: 2971]
GtoPdb Parasite growth inhibition assay - 7.49 pEC50 32 nM EC50 Nat Commun (2014) 5: 5521 [PMID:25422853]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.