repotrectinib [Ligand Id: 10316] activity data from GtoPdb
Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| neurotrophic receptor tyrosine kinase 1 in Human [GtoPdb: 1817] [UniProtKB: P04629] | ||||||||
| GtoPdb | - | - | 9.28 | pIC50 | 0.53 | nM | IC50 | Cancer Discov (2018) 8: 1227-1236 [PMID:30093503] |
| neurotrophic receptor tyrosine kinase 2 in Human [GtoPdb: 1818] [UniProtKB: Q16620] | ||||||||
| GtoPdb | - | - | 9.52 | pIC50 | 0.3 | nM | IC50 | Cancer Discov (2018) 8: 1227-1236 [PMID:30093503] |
| neurotrophic receptor tyrosine kinase 3 in Human [GtoPdb: 1819] [UniProtKB: Q16288] | ||||||||
| GtoPdb | - | - | 9.68 | pIC50 | 0.21 | nM | IC50 | Cancer Discov (2018) 8: 1227-1236 [PMID:30093503] |
| ALK receptor tyrosine kinase in Human [GtoPdb: 1839] [UniProtKB: Q9UM73] | ||||||||
| GtoPdb | - | - | 8.98 | pIC50 | 1.04 | nM | IC50 | Cancer Discov (2018) 8: 1227-1236 [PMID:30093503] |
| c-ros oncogene 1, receptor tyrosine kinase in Human [GtoPdb: 1840] [UniProtKB: P08922] | ||||||||
| GtoPdb | - | - | 10.15 | pIC50 | 0.07 | nM | IC50 | Cancer Discov (2018) 8: 1227-1236 [PMID:30093503] |
| Janus kinase 2 in Human [GtoPdb: 2048] [UniProtKB: O60674] | ||||||||
| GtoPdb | - | - | 8.98 | pIC50 | 1.04 | nM | IC50 | Cancer Discov (2018) 8: 1227-1236 [PMID:30093503] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
