SAR7334 [Ligand Id: 10283] activity data from GtoPdb

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  • TRPC3 in Human [GtoPdb: 488] [UniProtKB: Q13507]
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  • TRPC6 in Human [GtoPdb: 491] [UniProtKB: Q9Y210]
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  • TRPC7 in Human [GtoPdb: 492] [UniProtKB: Q9HCX4]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
TRPC3 in Human [GtoPdb: 488] [UniProtKB: Q13507]
GtoPdb - - 6.55 pIC50 282 nM IC50 Br J Pharmacol (2015) 172: 3650-60 [PMID:25847402]
TRPC6 in Human [GtoPdb: 491] [UniProtKB: Q9Y210]
GtoPdb - - 8.02 pIC50 9.5 nM IC50 Br J Pharmacol (2015) 172: 3650-60 [PMID:25847402]
TRPC7 in Human [GtoPdb: 492] [UniProtKB: Q9HCX4]
GtoPdb - - 6.65 pIC50 226 nM IC50 Br J Pharmacol (2015) 172: 3650-60 [PMID:25847402]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.