GSK1702934A [Ligand Id: 10278] activity data from GtoPdb

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  • TRPC3 in Human [GtoPdb: 488] [UniProtKB: Q13507]
Created with Highcharts 10.3.3ValuesChart context menuTRPC3pKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
  • TRPC6 in Human [GtoPdb: 491] [UniProtKB: Q9Y210]
Created with Highcharts 10.3.3ValuesChart context menuTRPC6pKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
TRPC3 in Human [GtoPdb: 488] [UniProtKB: Q13507]
GtoPdb Activation of hTRPC3-mediated currents in HEK293 cells in whole-cell patch-clamp experiments. - 7.1 pEC50 80 nM EC50 Biophys J (2013) 104: 454a
TRPC6 in Human [GtoPdb: 491] [UniProtKB: Q9Y210]
GtoPdb Activation of TRPC6-mediated currents in HEK293 cells in whole-cell patch-clamp experiments. - 6.36 pIC50 440 nM IC50 Biophys J (2013) 104: 454a

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.