UCT943 [Ligand Id: 10093] activity data from GtoPdb

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  • Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum V1/S [GtoPdb: 2972]
  • Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium berghei [GtoPdb: 2972]
  • Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium cynomolgi [GtoPdb: 2972]
  • Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum [GtoPdb: 2972]
  • Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum K1 [GtoPdb: 2972]
  • Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum NF54 [GtoPdb: 2972]
  • Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum 7G8 [GtoPdb: 2972]
  • Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum Dd2 [GtoPdb: 2972]
  • Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum HB3 [GtoPdb: 2972]
  • Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum D6 [GtoPdb: 2972]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum V1/S [GtoPdb: 2972]
GtoPdb Parasite growth inhibition assay - 8.38 pIC50 4.2 nM IC50 Antimicrob Agents Chemother (2018) 62: [PMID:29941635]
Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium berghei [GtoPdb: 2972]
GtoPdb Parasite liver stage assay - 9.04 pIC50 0.92 nM IC50 Antimicrob Agents Chemother (2018) 62: [PMID:29941635]
Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium cynomolgi [GtoPdb: 2972]
GtoPdb Parasite liver stage assay - 8 pIC50 <10 nM IC50 Antimicrob Agents Chemother (2018) 62: [PMID:29941635]
Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum [GtoPdb: 2972]
GtoPdb Parasite gametocyte viability assay - 6.87 pIC50 134 nM IC50 Antimicrob Agents Chemother (2018) 62: [PMID:29941635]
GtoPdb Standard membrane feeding assay (SMFA) - 7.02 pIC50 96 nM IC50 Antimicrob Agents Chemother (2018) 62: [PMID:29941635]
GtoPdb Parasite dual gamete formation assay (DGFA) - 7.1 pIC50 80 nM IC50 Antimicrob Agents Chemother (2018) 62: [PMID:29941635]
GtoPdb Parasite gametocyte viability assay - 7.18 pIC50 66 nM IC50 Antimicrob Agents Chemother (2018) 62: [PMID:29941635]
Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum K1 [GtoPdb: 2972]
GtoPdb Parasite growth inhibition assay - 8.33 pIC50 4.7 nM IC50 Antimicrob Agents Chemother (2018) 62: [PMID:29941635]
Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum NF54 [GtoPdb: 2972]
GtoPdb Parasite growth inhibition assay - 8.27 pIC50 5.4 nM IC50 Antimicrob Agents Chemother (2018) 62: [PMID:29941635]
Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum 7G8 [GtoPdb: 2972]
GtoPdb Parasite growth inhibition assay - 8.39 pIC50 4.1 nM IC50 Antimicrob Agents Chemother (2018) 62: [PMID:29941635]
Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum Dd2 [GtoPdb: 2972]
GtoPdb Parasite growth inhibition assay - 8.24 pIC50 5.7 nM IC50 Antimicrob Agents Chemother (2018) 62: [PMID:29941635]
Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum HB3 [GtoPdb: 2972]
GtoPdb Parasite growth inhibition assay - 8.43 pIC50 3.7 nM IC50 Antimicrob Agents Chemother (2018) 62: [PMID:29941635]
Plasmodium falciparum phosphatidylinositol 4-kinase beta in Plasmodium falciparum D6 [GtoPdb: 2972]
GtoPdb Parasite growth inhibition assay - 8.28 pIC50 5.2 nM IC50 Antimicrob Agents Chemother (2018) 62: [PMID:29941635]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.