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A list of approved drugs that modulate GABAA channel activity by binding to the allosteric benzodiazepine site. These drugs increase the inhibitory effects of GABA.
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            alprazolam
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            chlordiazepoxide
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            clobazam
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            clonazepam
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            clorazepate
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            diazepam
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            estazolam
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            eszopiclone
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            flumazenil
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            flunitrazepam
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            flurazepam
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            halazepam
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            lorazepam
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            lormetazepam
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            midazolam
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            oxazepam
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            quazepam
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            temazepam
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            triazolam
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            zaleplon
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            zolpidem
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Database page citation:
Benzodiazepine class drugs. Accessed on 31/10/2025. IUPHAR/BPS Guide to PHARMACOLOGY, http://www.guidetopharmacology.org/GRAC/FamilyDisplayForward?familyId=1072.